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TargetOxysterols receptor LXR-beta
LigandBDBM19992
Substrate/Competitorbiotinylated SRC-1 peptide
Meas. Tech.Cell-Free Ligand Sensing Assay (LiSA)-LXRbeta-SRC1 Assay
pH7.5±n/a
Temperature295.15±n/a K
EC50 20±10 nM
Citation Jaye, MCKrawiec, JACampobasso, NSmallwood, AQiu, CLu, QKerrigan, JJDe Los Frailes Alvaro, MLaffitte, BLiu, WSMarino, JPMeyer, CRNichols, JAParks, DJPerez, PSarov-Blat, LSeepersaud, SDSteplewski, KMThompson, SKWang, PWatson, MAWebb, CLHaigh, DCaravella, JAMacphee, CHWillson, TMCollins, JL Discovery of substituted maleimides as liver X receptor agonists and determination of a ligand-bound crystal structure. J Med Chem48:5419-22 (2005) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Oxysterols receptor LXR-beta
Name:Oxysterols receptor LXR-beta
Synonyms:LXRB | Liver X receptor beta (NR1H2) | Liver X, LXR beta | NER | NR1H2 | NR1H2_HUMAN | Nuclear receptor NER | UNR | Ubiquitously-expressed nuclear receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:50978.79
Organism:Homo sapiens (Human)
Description:P55055
Residue:460
Sequence:
MSSPTTSSLDTPLPGNGPPQPGAPSSSPTVKEEGPEPWPGGPDPDVPGTDEASSACSTDW
VIPDPEEEPERKRKKGPAPKMLGHELCRVCGDKASGFHYNVLSCEGCKGFFRRSVVRGGA
RRYACRGGGTCQMDAFMRRKCQQCRLRKCKEAGMREQCVLSEEQIRKKKIRKQQQESQSQ
SQSPVGPQGSSSSASGPGASPGGSEAGSQGSGEGEGVQLTAAQELMIQQLVAAQLQCNKR
SFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQI
ALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMR
RLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRM
LMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVHE
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  Blast E-value cutoff:
BDBM19992
biotinylated SRC-1 peptide
Name:biotinylated SRC-1 peptide
Synonyms:n/a
Type:Peptide
Mol. Mass.:3157.52
Organism:n/a
Description:A biotinylated peptide comprises amino acids 675-699 of steroid receptor coactivator 1 (SRC1).
Residue:28
Sequence:
CPSSHSSLTERHKILHRLLQEGSPS-CONH2