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TargetCaspase-6
LigandBDBM223
Substrate/CompetitorCaspase-6 Fluorometric Substrate Ac-Val-Glu-Ile-Asp-AFC
Meas. Tech.Fluorometric Assay
pH7.4±n/a
Temperature298.15±n/a K
Ki 190±n/a nM
Citation Choong, ICLew, WLee, DPham, PBurdett, MTLam, JWWiesmann, CLuong, TNFahr, BDeLano, WLMcDowell, RSAllen, DAErlanson, DAGordon, EMO'Brien, T Identification of potent and selective small-molecule inhibitors of caspase-3 through the use of extended tethering and structure-based drug design. J Med Chem45:5005-22 (2002) [PubMed]  Article
More Info.:Get all data from this article,  Inhibition_Run data,   Solution Info,  Assay Method
 
Caspase-6
Name:Caspase-6
Synonyms:Apoptotic protease Mch-2 | CASP-6 | CASP6 | CASP6_HUMAN | Caspase | MCH2
Type:Enzyme
Mol. Mass.:33312.62
Organism:Homo sapiens (Human)
Description:P55212
Residue:293
Sequence:
MSSASGLRRGHPAGGEENMTETDAFYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLT
LPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLS
HGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQACRGNQHDVPVIPLDVVDN
QTEKLDTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYG
SSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKSN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM223
Caspase-6 Fluorometric Substrate Ac-Val-Glu-Ile-Asp-AFC
Name:Caspase-6 Fluorometric Substrate Ac-Val-Glu-Ile-Asp-AFC
Synonyms:n/a
Type:Peptide
Mol. Mass.:472.49
Organism:n/a
Description:Molecular Mass of VEID
Residue:4
Sequence:
VEID