Reaction Details |
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Target | Aurora kinase B |
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Ligand | BDBM26303 |
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Substrate/Competitor | Biotinylated Peptide Substrate |
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Meas. Tech. | Aurora B Kinase Inhibition Assay |
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pH | 7.5±n/a |
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Temperature | 295.15±n/a K |
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Ki | <1±n/a nM |
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Citation | Foote, KM; Mortlock, AA; Heron, NM; Jung, FH; Hill, GB; Pasquet, G; Brady, MC; Green, S; Heaton, SP; Kearney, S; Keen, NJ; Odedra, R; Wedge, SR; Wilkinson, RW Synthesis and SAR of 1-acetanilide-4-aminopyrazole-substituted quinazolines: selective inhibitors of Aurora B kinase with potent anti-tumor activity. Bioorg Med Chem Lett18:1904-9 (2008) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Aurora kinase B |
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Name: | Aurora kinase B |
Synonyms: | AIK2 | AIM-1 | AIM1 | AIRK2 | ARK2 | AURKB | AURKB_HUMAN | Aurora B kinase (aurB) | Aurora B-INCENP | Aurora kinase 2 | Aurora kinase B (AURKB) | Aurora-related kinase 2 | STK-1 | STK1 | STK12 | STK5 | Serine/threonine-protein kinase aurora B |
Type: | Protein |
Mol. Mass.: | 39327.72 |
Organism: | Homo sapiens (Human) |
Description: | Q96GD4 |
Residue: | 344 |
Sequence: | MAQKENSYPWPYGRQTAPSGLSTLPQRVLRKEPVTPSALVLMSRSNVQPTAAPGQKVMEN
SSGTPDILTRHFTIDDFEIGRPLGKGKFGNVYLAREKKSHFIVALKVLFKSQIEKEGVEH
QLRREIEIQAHLHHPNILRLYNYFYDRRRIYLILEYAPRGELYKELQKSCTFDEQRTATI
MEELADALMYCHGKKVIHRDIKPENLLLGLKGELKIADFGWSVHAPSLRRKTMCGTLDYL
PPEMIEGRMHNEKVDLWCIGVLCYELLVGNPPFESASHNETYRRIVKVDLKFPASVPMGA
QDLISKLLRHNPSERLPLAQVSAHPWVRANSRRVLPPSALQSVA
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BDBM26303 |
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Biotinylated Peptide Substrate |
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Name: | Biotinylated Peptide Substrate |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 2374.22 |
Organism: | n/a |
Description: | n/a |
Residue: | 20 |
Sequence: | biotinyl-Ahx-tetra(LRRWSLG)
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