Reaction Details |
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Target | KiSS-1 receptor |
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Ligand | BDBM26345 |
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Substrate/Competitor | [125I]Kisspeptin-15 |
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Meas. Tech. | Receptor Binding Assay |
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pH | 7.3±n/a |
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Temperature | 298.15±n/a K |
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IC50 | 5.7±n/a nM |
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Citation | Tomita, K; Oishi, S; Ohno, H; Peiper, SC; Fujii, N Development of Novel G-Protein-Coupled Receptor 54 Agonists with Resistance to Degradation by Matrix Metalloproteinase. J Med Chem51:7645-9 (2008) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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KiSS-1 receptor |
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Name: | KiSS-1 receptor |
Synonyms: | AXOR12 | G-protein Coupled Receptor 54 | G-protein coupled receptor 54 (GPR54) | GPR54 | Hypogonadotropin-1 | KISS1R | KISSR_HUMAN | KiSS-1R | Kisspeptins receptor | Metastin receptor | hOT7T175 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 42613.79 |
Organism: | Homo sapiens (Human) |
Description: | Binding assay was performed using membranes from the CHO cell transfectants. |
Residue: | 398 |
Sequence: | MHTVATSGPNASWGAPANASGCPGCGANASDGPVPSPRAVDAWLVPLFFAALMLLGLVGN
SLVIYVICRHKPMRTVTNFYIANLAATDVTFLLCCVPFTALLYPLPGWVLGDFMCKFVNY
IQQVSVQATCATLTAMSVDRWYVTVFPLRALHRRTPRLALAVSLSIWVGSAAVSAPVLAL
HRLSPGPRAYCSEAFPSRALERAFALYNLLALYLLPLLATCACYAAMLRHLGRVAVRPAP
ADSALQGQVLAERAGAVRAKVSRLVAAVVLLFAACWGPIQLFLVLQALGPAGSWHPRSYA
AYALKTWAHCMSYSNSALNPLLYAFLGSHFRQAFRRVCPCAPRRPRRPRRPGPSDPAAPH
AELLRLGSHPAPARAQKPGSSGLAARGLCVLGEDNAPL
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BDBM26345 |
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[125I]Kisspeptin-15 |
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Name: | [125I]Kisspeptin-15 |
Synonyms: | n/a |
Type: | radiolabeled peptide |
Mol. Mass.: | 1872.07 |
Organism: | n/a |
Description: | n/a |
Residue: | 15 |
Sequence: | |