| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM29093 |
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| Substrate/Competitor | BDBM21244 |
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| Meas. Tech. | CB Receptor Radioligand Binding Assay (Ki) |
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| Ki | 2420±n/a nM |
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| Citation |  Appendino, G; Ligresti, A; Minassi, A; Cascio, MG; Allarà, M; Taglialatela-Scafati, O; Pertwee, RG; De Petrocellis, L; Di Marzo, V Conformationally constrained fatty acid ethanolamides as cannabinoid and vanilloid receptor probes. J Med Chem52:3001-9 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM29093 |
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| BDBM21244 |
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| Name | BDBM29093 |
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| Synonyms: | cyclopropanolamide, 11b |
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| Type | Small organic molecule |
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| Emp. Form. | C21H39NO2 |
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| Mol. Mass. | 337.5399 |
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| SMILES | CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H]1C[C@@H]1O |r| |
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| Structure | 
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