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TargetBcl-2-like protein 1
LigandBDBM31419
Substrate/CompetitorFl-Bak peptide
Meas. Tech.Fluorescence Polarization Assay
pH7.4±n/a
Temperature298.15±n/a K
Ki 4820±n/a nM
Citation Yin, HLee, GISedey, KAKutzki, OPark, HSOrner, BPErnst, JTWang, HGSebti, SMHamilton, AD Terphenyl-Based Bak BH3 alpha-helical proteomimetics as low-molecular-weight antagonists of Bcl-xL. J Am Chem Soc127:10191-6 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Inhibition_Run data,   Solution Info,  Assay Method
 
Bcl-2-like protein 1
Name:Bcl-2-like protein 1
Synonyms:Anti-apoptotic Bcl-2 protein | Apoptosis Regulator Bcl-xL | Apoptosis regulator Bcl-X | B2CL1_HUMAN | BCL2-like 1 isoform 1 | BCL2L | BCL2L1 | BCLX | Bcl-2-like protein 1 (Bcl-XL) | Bcl-X | Bcl-xL/Bcl-2-binding component 3 | Bcl2-L-1 | Bcl2-antagonist of cell death (BAD)
Type:Mitochondrion membrane; Single-pass membrane protein
Mol. Mass.:26039.60
Organism:Homo sapiens (Human)
Description:n/a
Residue:233
Sequence:
MSQSNRELVVDFLSYKLSQKGYSWSQFSDVEENRTEAPEGTESEMETPSAINGNPSWHLA
DSPAVNGATGHSSSLDAREVIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAY
QSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEP
WIQENGGWDTFVELYGNNAAAESRKGQERFNRWFLTGMTVAGVVLLGSLFSRK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM31419
Fl-Bak peptide
Name:Fl-Bak peptide
Synonyms:n/a
Type:Fluoroscein-labled peptide
Mol. Mass.:2079.80
Organism:n/a
Description:The N-terminus of fluoroscein-labled Bak peptide was capped with the fluorophore and the C-terminus was amidated.
Residue:19
Sequence:
GQVGRQLAIIGDDINR-CONH2