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TargetIsoform Bcl-X(L) of Bcl-2-like protein 1 (Bcl-xL)
LigandBDBM32280
Substrate/CompetitorF-Bim
Meas. Tech.Multiplexed dose response screen for small molecule regulators of Bcl-2 family protein interactions, specifically Bim-Bcl-XL.
pH7.4±n/a
Temperature277.15±n/a K
EC50 23130±n/a nM
Citation PubChem, PC Multiplexed dose response screen for small molecule regulators of Bcl-2 family protein interactions, specifically Bim-Bcl-XL. PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Isoform Bcl-X(L) of Bcl-2-like protein 1 (Bcl-xL)
Name:Isoform Bcl-X(L) of Bcl-2-like protein 1 (Bcl-xL)
Synonyms:B-cell lymphoma-extra large protein (Bcl-xL) | B2CL1_HUMAN | BCL-xL | BCL2L | BCL2L1 | BCLX | Bcl-2-like protein 1 (Bcl-xL) | Isoform Bcl-X(L)
Type:Homodimers/heterodimers with BAX, BAK and BCL2
Mol. Mass.:26053.63
Organism:Homo sapiens (Human)
Description:gi_510901
Residue:233
Sequence:
MSQSNRELVVDFLSYKLSQKGYSWSQFSDVEENRTEAPEGTESEMETPSAINGNPSWHLA
DSPAVNGATAHSSSLDAREVIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAY
QSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEP
WIQENGGWDTFVELYGNNAAAESRKGQERFNRWFLTGMTVAGVVLLGSLFSRK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM32280
F-Bim
Name:F-Bim
Synonyms:n/a
Type:fluorescent peptide probe
Mol. Mass.:3923.40
Organism:n/a
Description:n/a
Residue:32
Sequence:
FITC-Ahx-DMRPEIWIAQELRRIGDEFNAYYAR-OH