Reaction Details |
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Target | Sliding-clamp-loader large/small subunit |
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Ligand | BDBM36318 |
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Substrate/Competitor | BDBM50118233 |
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Meas. Tech. | colorimetric ATPase assay |
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pH | 7.5±0 |
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Temperature | 298.15±0 K |
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Ki | 3.7e+4± 8e+3 nM |
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Citation | Eng, K; Scouten-Ponticelli, SK; Sutton, M; Berdis, A Selective Inhibition of DNA Replicase Assembly by a Non-natural Nucleotide: Exploiting the Structural Diversity of ATP-Binding Sites ACS Chem Biol5:183-94 (2010) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Sliding-clamp-loader large/small subunit |
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Name: | Sliding-clamp-loader large/small subunit |
Synonyms: | ATP-dependent clamp loaders gp44/62 |
Type: | n/a |
Mol. Mass.: | n/a |
Description: | n/a |
Components: | This complex has 2 components. |
Component 1 |
Name: | Sliding-clamp-loader large subunit |
Synonyms: | 44 | Clamp loader large subunit | Gene product 44 | LOADL_BPT4 | Sliding-clamp-loader gp44 subunit | gp44 |
Type: | n/a |
Mol. Mass.: | 35788.87 |
Organism: | Enterobacteria phage T4 (Bacteriophage T4) |
Description: | P04526 |
Residue: | 319 |
Sequence: | MITVNEKEHILEQKYRPSTIDECILPAFDKETFKSITSKGKIPHIILHSPSPGTGKTTVA
KALCHDVNADMMFVNGSDCKIDFVRGPLTNFASAASFDGRQKVIVIDEFDRSGLAESQRH
LRSFMEAYSSNCSIIITANNIDGIIKPLQSRCRVITFGQPTDEDKIEMMKQMIRRLTEIC
KHEGIAIADMKVVAALVKKNFPDFRKTIGELDSYSSKGVLDAGILSLVTNDRGAIDDVLE
SLKNKDVKQLRALAPKYAADYSWFVGKLAEEIYSRVTPQSIIRMYEIVGENNQYHGIAAN
TELHLAYLFIQLACEMQWK
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Component 2 |
Name: | Sliding-clamp-loader small subunit |
Synonyms: | 62 | Clamp loader small subunit | Gene product 62 | LOADS_BPT4 | Sliding-clamp-loader gp44 subunit | gp62 |
Type: | n/a |
Mol. Mass.: | 21366.49 |
Organism: | Enterobacteria phage T4 (Bacteriophage T4) |
Description: | P04527 |
Residue: | 187 |
Sequence: | MSLFKDDIQLNEHQVAWYSKDWTAVQSAADSFKEKAENEFFEIIGAINNKTKCSIAQKDY
SKFMVENALSQFPECMPAVYAMNLIGSGLSDEAHFNYLMAAVPRGKRYGKWAKLVEDSTE
VLIIKLLAKRYQVNTNDAINYKSILTKNGKLPLVLKELKGLVTDDFLKEVTKNVKEQKQL
KKLALEW
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BDBM36318 |
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BDBM50118233 |
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Name | BDBM36318 |
Synonyms: | 5-carboxylate-indolyl- 2'-deoxyriboside triphosphate | 5-cyclohexyl-indolyl- 2'-deoxyriboside triphosphate | d5-CITP |
Type | Small organic molecule |
Emp. Form. | C14H18NO14P3 |
Mol. Mass. | 517.2123 |
SMILES | [H][C@]1(O)C[C@@]([H])(O[C@]1([H])COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1ccc2cc(ccc12)C(O)=O |
Structure |
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