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TargetDNA polymerase III subunit tau
LigandBDBM36314
Substrate/CompetitorBDBM50118233
Meas. Tech.colorimetric ATPase assay
pH7.5±0
Temperature310.15±0 K
Ki 4.50e+4± 1.85e+4 nM
Citation Eng, KScouten-Ponticelli, SKSutton, MBerdis, A Selective Inhibition of DNA Replicase Assembly by a Non-natural Nucleotide: Exploiting the Structural Diversity of ATP-Binding Sites ACS Chem Biol5:183-94 (2010) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
DNA polymerase III subunit tau
Name:DNA polymerase III subunit tau
Synonyms:ATP-dependent clamp loader gamma -complex | DNA polymerase III subunit gamma | DPO3X_ECOLI | dnaX | dnaZ | dnaZX
Type:PROTEIN
Mol. Mass.:71139.93
Organism:Escherichia coli
Description:P06710
Residue:643
Sequence:
MSYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAK
GLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRF
KVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDV
EQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAM
LGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPA
ALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFH
PRMPLPEPEVPRQSFAPVAPTAVMTPTQVPPQPQSAPQQAPTVPLPETTSQVLAARQQLQ
RVQGATKAKKSEPAAATRARPVNNAALERLASVTDRVQARPVPSALEKAPAKKEAYRWKA
TTPVMQQKEVVATPKALKKALEHEKTPELAAKLAAEAIERDPWAAQVSQLSLPKLVEQVA
LNAWKEESDNAVCLHLRSSQRHLNNRGAQQKLAEALSMLKGSTVELTIVEDDNPAVRTPL
EWRQAIYEEKLAQARESIIADNNIQTLRRFFDAELDEESIRPI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM36314
BDBM50118233
NameBDBM36314
Synonyms:5-amino-indolyl- 2'-deoxyriboside triphosphate | d5-AITP
TypeSmall organic molecule
Emp. Form.C13H19N2O12P3
Mol. Mass.488.2174
SMILES[H][C@]1(O)C[C@@]([H])(O[C@]1([H])COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1ccc2cc(N)ccc12
Structure
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