Reaction Details |
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Target | DNA polymerase III subunit tau |
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Ligand | BDBM36314 |
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Substrate/Competitor | BDBM50118233 |
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Meas. Tech. | colorimetric ATPase assay |
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pH | 7.5±0 |
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Temperature | 310.15±0 K |
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Ki | 4.50e+4± 1.85e+4 nM |
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Citation | Eng, K; Scouten-Ponticelli, SK; Sutton, M; Berdis, A Selective Inhibition of DNA Replicase Assembly by a Non-natural Nucleotide: Exploiting the Structural Diversity of ATP-Binding Sites ACS Chem Biol5:183-94 (2010) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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DNA polymerase III subunit tau |
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Name: | DNA polymerase III subunit tau |
Synonyms: | ATP-dependent clamp loader gamma -complex | DNA polymerase III subunit gamma | DPO3X_ECOLI | dnaX | dnaZ | dnaZX |
Type: | PROTEIN |
Mol. Mass.: | 71139.93 |
Organism: | Escherichia coli |
Description: | P06710 |
Residue: | 643 |
Sequence: | MSYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAK
GLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRF
KVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDV
EQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAM
LGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPA
ALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFH
PRMPLPEPEVPRQSFAPVAPTAVMTPTQVPPQPQSAPQQAPTVPLPETTSQVLAARQQLQ
RVQGATKAKKSEPAAATRARPVNNAALERLASVTDRVQARPVPSALEKAPAKKEAYRWKA
TTPVMQQKEVVATPKALKKALEHEKTPELAAKLAAEAIERDPWAAQVSQLSLPKLVEQVA
LNAWKEESDNAVCLHLRSSQRHLNNRGAQQKLAEALSMLKGSTVELTIVEDDNPAVRTPL
EWRQAIYEEKLAQARESIIADNNIQTLRRFFDAELDEESIRPI
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BDBM36314 |
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BDBM50118233 |
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Name | BDBM36314 |
Synonyms: | 5-amino-indolyl- 2'-deoxyriboside triphosphate | d5-AITP |
Type | Small organic molecule |
Emp. Form. | C13H19N2O12P3 |
Mol. Mass. | 488.2174 |
SMILES | [H][C@]1(O)C[C@@]([H])(O[C@]1([H])COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1ccc2cc(N)ccc12 |
Structure |
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