Reaction Details |
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Target | Receptor protein serine/threonine kinase |
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Ligand | BDBM5416 |
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Substrate/Competitor | poly(Glu4, Tyr) |
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Meas. Tech. | Kinase assay Dorsalization |
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EC50 | 1e+3±n/a nM |
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Citation | Hao, J; Ho, JN; Lewis, JA; Karim, KA; Daniels, RN; Gentry, PR; Hopkins, CR; Lindsley, CW; Hong, CC In vivo structure-activity relationship study of dorsomorphin analogues identifies selective VEGF and BMP inhibitors. ACS Chem Biol5:245-53 (2010) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Receptor protein serine/threonine kinase |
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Name: | Receptor protein serine/threonine kinase |
Synonyms: | B3DJG0 | BMP | Bmpr1a protein | Bone morphogenetic protein |
Type: | n/a |
Mol. Mass.: | 59502.00 |
Organism: | Danio rerio (Zebrafish) |
Description: | B3DJG0 |
Residue: | 526 |
Sequence: | MRQLLFITVVLTGVCLLLTLCSGGQNPDHVLQGTGVKLDSRRPGDDSTIAPEDAARFLSC
HCSGHCPDDAKNNTCETNGQCFAIIEEDENGDVILSSGCMKYEGSHFQCKDSQFAQTRRT
IECCQFDFCNQDLKPELPPRDSEPPDPHWLAFLISVTVCFCALICVTVICYYRYKWQTER
QRYHRDLEQDEAFIPAGESLKDLINQSQTSGSGSGLPLLVQRTIAKQIQTVRMIGKGRYG
EVWLGRWRGEKVAVKVFFTREEASWFRETEIYQTVLMRHENILGFIAADINGTGASTQLY
LITDYHENGSLYDYLKFTTLDTQALLRLAFSAACGLCHLHTEIYGTQGKPAIAHRDLKSK
NILIKKNGTCCIADLGLAVKFNSDTNEVDLPLSTRMGTRRYMAPEVLDETLNKNHFQAYI
MADIYSYGLVIWEMARRCVTGGIVEEYQLPYYEMVPSDPSYEDMLEVVCVKGLRPTVSNR
WNSDECLRAMLKLMSECWAHNPASRLTILRVKKTLAKMVESQDIKI
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BDBM5416 |
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poly(Glu4, Tyr) |
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Name: | poly(Glu4, Tyr) |
Synonyms: | n/a |
Type: | Random copolymer |
Mol. Mass.: | 358.43 |
Organism: | n/a |
Description: | n/a |
Residue: | 3 |
Sequence: | |