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TargetReceptor protein serine/threonine kinase
LigandBDBM36356
Substrate/Competitorpoly(Glu4, Tyr)
Meas. Tech.Kinase assay Dorsalization
EC50 1e+3±n/a nM
Citation Hao, JHo, JNLewis, JAKarim, KADaniels, RNGentry, PRHopkins, CRLindsley, CWHong, CC In vivo structure-activity relationship study of dorsomorphin analogues identifies selective VEGF and BMP inhibitors. ACS Chem Biol5:245-53 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Receptor protein serine/threonine kinase
Name:Receptor protein serine/threonine kinase
Synonyms:B3DJG0 | BMP | Bmpr1a protein | Bone morphogenetic protein
Type:n/a
Mol. Mass.:59502.00
Organism:Danio rerio (Zebrafish)
Description:B3DJG0
Residue:526
Sequence:
MRQLLFITVVLTGVCLLLTLCSGGQNPDHVLQGTGVKLDSRRPGDDSTIAPEDAARFLSC
HCSGHCPDDAKNNTCETNGQCFAIIEEDENGDVILSSGCMKYEGSHFQCKDSQFAQTRRT
IECCQFDFCNQDLKPELPPRDSEPPDPHWLAFLISVTVCFCALICVTVICYYRYKWQTER
QRYHRDLEQDEAFIPAGESLKDLINQSQTSGSGSGLPLLVQRTIAKQIQTVRMIGKGRYG
EVWLGRWRGEKVAVKVFFTREEASWFRETEIYQTVLMRHENILGFIAADINGTGASTQLY
LITDYHENGSLYDYLKFTTLDTQALLRLAFSAACGLCHLHTEIYGTQGKPAIAHRDLKSK
NILIKKNGTCCIADLGLAVKFNSDTNEVDLPLSTRMGTRRYMAPEVLDETLNKNHFQAYI
MADIYSYGLVIWEMARRCVTGGIVEEYQLPYYEMVPSDPSYEDMLEVVCVKGLRPTVSNR
WNSDECLRAMLKLMSECWAHNPASRLTILRVKKTLAKMVESQDIKI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM36356
poly(Glu4, Tyr)
Name:poly(Glu4, Tyr)
Synonyms:n/a
Type:Random copolymer
Mol. Mass.:358.43
Organism:n/a
Description:n/a
Residue:3
Sequence:
n/a