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TargetfMet-Leu-Phe receptor
LigandBDBM37628
Substrate/Competitorn/a
Meas. Tech.Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki 8900±n/a nM
Citation PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
fMet-Leu-Phe receptor
Name:fMet-Leu-Phe receptor
Synonyms:FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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  Blast E-value cutoff:
BDBM37628
n/a
NameBDBM37628
Synonyms:1-Benzyl-4-(furan-2-carbonyl)-3-hydroxy-5-pyridin-4-yl-1,5-dihydro-pyrrol-2-one | 1-benzyl-3-(furan-2-carbonyl)-4-hydroxy-2-pyridin-4-yl-2H-pyrrol-5-one | 1-benzyl-4-(2-furoyl)-3-hydroxy-5-(4-pyridyl)-3-pyrrolin-2-one | 3-(furan-2-ylcarbonyl)-4-oxidanyl-1-(phenylmethyl)-2-pyridin-4-yl-2H-pyrrol-5-one | 3-[2-furanyl(oxo)methyl]-4-hydroxy-1-(phenylmethyl)-2-pyridin-4-yl-2H-pyrrol-5-one | MLS000034860 | SMR000013491 | cid_655756
TypeSmall organic molecule
Emp. Form.C21H16N2O4
Mol. Mass.360.3627
SMILESO=C(C1C(N(Cc2ccccc2)C(=O)C1=O)c1ccncc1)c1ccco1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: