| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 1 |
|---|
| Ligand | BDBM31040 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing |
|---|
| IC50 | 1185±n/a nM |
|---|
| Citation |  PubChem, PC In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing PubChem Bioassay(2006)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Dual specificity protein phosphatase 1 |
|---|
| Name: | Dual specificity protein phosphatase 1 |
|---|
| Synonyms: | CL100 | DUS1_HUMAN | DUSP1 | Dual specificity protein phosphatase hVH1 | MAP kinase phosphatase 1 | MKP-1 | MKP1 | PTPN10 | Protein-tyrosine phosphatase CL100 | VH1 |
|---|
| Type: | Protein phosphatase |
|---|
| Mol. Mass.: | 39301.48 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_4758204 |
|---|
| Residue: | 367 |
|---|
| Sequence: | MVMEVGTLDAGGLRALLGERAAQCLLLDCRSFFAFNAGHIAGSVNVRFSTIVRRRAKGAM
GLEHIVPNAELRGRLLAGAYHAVVLLDERSAALDGAKRDGTLALAAGALCREARAAQVFF
LKGGYEAFSASCPELCSKQSTPMGLSLPLSTSVPDSAESGCSSCSTPLYDQGGPVEILPF
LYLGSAYHASRKDMLDALGITALINVSANCPNHFEGHYQYKSIPVEDNHKADISSWFNEA
IDFIDSIKNAGGRVFVHCQAGISRSATICLAYLMRTNRVKLDEAFEFVKQRRSIISPNFS
FMGQLLQFESQVLAPHCSAEAGSPAMAVLDRGTSTTTVFNFPVSIPVHSTNSALSYLQSP
ITTSPSC
|
|
|
|---|
| BDBM31040 |
|---|
| n/a |
|---|
| Name | BDBM31040 |
|---|
| Synonyms: | 1-Ethyl-6-methyl-3-phenyl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1-ethyl-6-methyl-3-phenyl-pyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1-ethyl-6-methyl-3-phenyl-pyrimido[5,4-e][1,2,4]triazine-5,7-quinone | 1-ethyl-6-methyl-3-phenylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | MLS000027832 | SMR000008919 | US9073941, 602 | cid_647501 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C14H13N5O2 |
|---|
| Mol. Mass. | 283.2853 |
|---|
| SMILES | CCn1nc(nc2c1nc(=O)n(C)c2=O)-c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
