| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 1 |
|---|
| Ligand | BDBM32102 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing |
|---|
| IC50 | 743±n/a nM |
|---|
| Citation |  PubChem, PC In vitro MKP-1 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing PubChem Bioassay(2006)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Dual specificity protein phosphatase 1 |
|---|
| Name: | Dual specificity protein phosphatase 1 |
|---|
| Synonyms: | CL100 | DUS1_HUMAN | DUSP1 | Dual specificity protein phosphatase hVH1 | MAP kinase phosphatase 1 | MKP-1 | MKP1 | PTPN10 | Protein-tyrosine phosphatase CL100 | VH1 |
|---|
| Type: | Protein phosphatase |
|---|
| Mol. Mass.: | 39301.48 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_4758204 |
|---|
| Residue: | 367 |
|---|
| Sequence: | MVMEVGTLDAGGLRALLGERAAQCLLLDCRSFFAFNAGHIAGSVNVRFSTIVRRRAKGAM
GLEHIVPNAELRGRLLAGAYHAVVLLDERSAALDGAKRDGTLALAAGALCREARAAQVFF
LKGGYEAFSASCPELCSKQSTPMGLSLPLSTSVPDSAESGCSSCSTPLYDQGGPVEILPF
LYLGSAYHASRKDMLDALGITALINVSANCPNHFEGHYQYKSIPVEDNHKADISSWFNEA
IDFIDSIKNAGGRVFVHCQAGISRSATICLAYLMRTNRVKLDEAFEFVKQRRSIISPNFS
FMGQLLQFESQVLAPHCSAEAGSPAMAVLDRGTSTTTVFNFPVSIPVHSTNSALSYLQSP
ITTSPSC
|
|
|
|---|
| BDBM32102 |
|---|
| n/a |
|---|
| Name | BDBM32102 |
|---|
| Synonyms: | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone | MLS000087831 | SMR000024051 | US9284299, PKF118-310 | US9738628, Compound PKF118-310 | cid_66541 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C7H7N5O2 |
|---|
| Mol. Mass. | 193.1628 |
|---|
| SMILES | Cn1ncnc2c1nc(=O)n(C)c2=O |
|---|
| Structure | 
|
|---|
Search and Browse
