Reaction Details |
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Target | N-formyl peptide receptor 2 |
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Ligand | BDBM40414 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1) |
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Ki | >40300±n/a nM |
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Citation | PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1) PubChem Bioassay(2007)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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N-formyl peptide receptor 2 |
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Name: | N-formyl peptide receptor 2 |
Synonyms: | ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 38968.35 |
Organism: | Homo sapiens (Human) |
Description: | P25090 |
Residue: | 351 |
Sequence: | METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVT
TICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIA
LDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNF
ASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPL
RVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPM
LYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
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BDBM40414 |
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n/a |
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Name | BDBM40414 |
Synonyms: | 3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(4-morpholinylmethyl)-2-(trifluoromethyl)-1-benzopyran-4-one | 3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(morpholin-4-ylmethyl)-2-(trifluoromethyl)chromen-4-one | 3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(morpholinomethyl)-2-(trifluoromethyl)chromone | 3-(3,4-dimethoxyphenyl)-8-(morpholin-4-ylmethyl)-7-oxidanyl-2-(trifluoromethyl)chromen-4-one | UNM000003540001 | cid_5449443 |
Type | Small organic molecule |
Emp. Form. | C23H22F3NO6 |
Mol. Mass. | 465.4191 |
SMILES | COc1ccc(cc1OC)-c1c(oc2c(CN3CCOCC3)c(O)ccc2c1=O)C(F)(F)F |
Structure |
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