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Reaction Details
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TargetN-formyl peptide receptor 2
LigandBDBM40414
Substrate/Competitorn/a
Meas. Tech.Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)
Ki>40300±n/a nM
Citation PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)  PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
N-formyl peptide receptor 2
Name:N-formyl peptide receptor 2
Synonyms:ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:38968.35
Organism:Homo sapiens (Human)
Description:P25090
Residue:351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVT
TICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIA
LDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNF
ASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPL
RVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPM
LYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
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  Blast E-value cutoff:
BDBM40414
n/a
NameBDBM40414
Synonyms:3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(4-morpholinylmethyl)-2-(trifluoromethyl)-1-benzopyran-4-one | 3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(morpholin-4-ylmethyl)-2-(trifluoromethyl)chromen-4-one | 3-(3,4-dimethoxyphenyl)-7-hydroxy-8-(morpholinomethyl)-2-(trifluoromethyl)chromone | 3-(3,4-dimethoxyphenyl)-8-(morpholin-4-ylmethyl)-7-oxidanyl-2-(trifluoromethyl)chromen-4-one | UNM000003540001 | cid_5449443
TypeSmall organic molecule
Emp. Form.C23H22F3NO6
Mol. Mass.465.4191
SMILESCOc1ccc(cc1OC)-c1c(oc2c(CN3CCOCC3)c(O)ccc2c1=O)C(F)(F)F
Structure
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