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Reaction Details
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TargetfMet-Leu-Phe receptor
LigandBDBM40411
Substrate/Competitorn/a
Meas. Tech.Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay
Ki 6000±n/a nM
Citation PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
fMet-Leu-Phe receptor
Name:fMet-Leu-Phe receptor
Synonyms:FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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BDBM40411
n/a
NameBDBM40411
Synonyms:(4E)-5-(2,5-dimethoxyphenyl)-4-[hydroxy(phenyl)methylene]-1-(3-pyridyl)pyrrolidine-2,3-quinone | (4E)-5-(2,5-dimethoxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-(3-pyridinyl)pyrrolidine-2,3-dione | (4E)-5-(2,5-dimethoxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-pyridin-3-ylpyrrolidine-2,3-dione | (4E)-5-(2,5-dimethoxyphenyl)-4-[oxidanyl(phenyl)methylidene]-1-pyridin-3-yl-pyrrolidine-2,3-dione | UNM000003538701 | cid_5291451
TypeSmall organic molecule
Emp. Form.C24H20N2O5
Mol. Mass.416.426
SMILESCOc1ccc(OC)c(c1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1c1cccnc1
Structure
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