Ki Summary

Reaction Details

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Target

fMet-Leu-Phe receptor

Ligand

BDBM40415

Substrate/Competitor

n/a

Meas. Tech.

Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay

2500±n/a nM

Citation

PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay PubChem Bioassay(2007)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

fMet-Leu-Phe receptor

Name:

fMet-Leu-Phe receptor

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

38456.14

Organism:

Homo sapiens (Human)

Description:

gi_4503779

Residue:

350

Sequence:

METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK

BDBM40415

n/a

Name

BDBM40415

Synonyms:

2-furancarboxylic acid [3-(2-chlorophenyl)-4-oxo-2-(trifluoromethyl)-1-benzopyran-7-yl] ester | UNM000003546901 | [3-(2-chlorophenyl)-4-oxidanylidene-2-(trifluoromethyl)chromen-7-yl] furan-2-carboxylate | [3-(2-chlorophenyl)-4-oxo-2-(trifluoromethyl)chromen-7-yl] furan-2-carboxylate | cid_1036526 | furan-2-carboxylic acid [3-(2-chlorophenyl)-4-keto-2-(trifluoromethyl)chromen-7-yl] ester

Type

Small organic molecule

Emp. Form.

C21H10ClF3O5

Mol. Mass.

434.749

SMILES

FC(F)(F)c1oc2cc(OC(=O)c3ccco3)ccc2c(=O)c1-c1ccccc1Cl |(4.41,2.51,;5.75,1.74,;6.52,3.08,;4.98,.41,;7.08,.97,;8.41,1.74,;9.75,.97,;11.13,1.8,;12.52,1,;13.85,1.78,;15.19,1.01,;15.19,-.53,;16.52,1.79,;17.93,1.17,;18.95,2.32,;18.18,3.65,;16.67,3.32,;12.52,-.6,;11.13,-1.39,;9.75,-.57,;8.41,-1.34,;8.41,-2.88,;7.08,-.57,;5.75,-1.34,;4.41,-.57,;3.08,-1.34,;3.08,-2.88,;4.41,-3.65,;5.75,-2.88,;7.08,-3.65,)|

Structure