| Reaction Details |
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 | Report a problem with these data |
| Target | fMet-Leu-Phe receptor |
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| Ligand | BDBM40419 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay |
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| Ki | 3400±n/a nM |
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| Citation |  PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| fMet-Leu-Phe receptor |
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| Name: | fMet-Leu-Phe receptor |
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| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38456.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4503779 |
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| Residue: | 350 |
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| Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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| BDBM40419 |
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| n/a |
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| Name | BDBM40419 |
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| Synonyms: | (4E)-5-(2,4-dimethoxyphenyl)-1-(3-imidazol-1-ylpropyl)-4-[oxidanyl(phenyl)methylidene]pyrrolidine-2,3-dione | (4E)-5-(2,4-dimethoxyphenyl)-4-[hydroxy(phenyl)methylene]-1-(3-imidazol-1-ylpropyl)pyrrolidine-2,3-quinone | (4E)-5-(2,4-dimethoxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-(3-imidazol-1-ylpropyl)pyrrolidine-2,3-dione | (4E)-5-(2,4-dimethoxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-[3-(1-imidazolyl)propyl]pyrrolidine-2,3-dione | UNM000003552201 | cid_5941053 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H25N3O5 |
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| Mol. Mass. | 447.4831 |
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| SMILES | COc1ccc(C2C(C(=O)c3ccccc3)C(=O)C(=O)N2CCCn2ccnc2)c(OC)c1 |
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| Structure | 
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