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TargetHematopoietic protein-tyrosine phosphatase (HEPTP)
LigandBDBM46207
Substrate/Competitorn/a
Meas. Tech.Fluorescent secondary assay for dose-response confirmation of chemical inhibitors of HePTP
IC50 274±n/a nM
Citation PubChem PC Fluorescent secondary assay for dose-response confirmation of chemical inhibitors of HePTP PubChem Bioassay (2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Hematopoietic protein-tyrosine phosphatase (HEPTP)
Name:Hematopoietic protein-tyrosine phosphatase (HEPTP)
Synonyms:He-PTP | Hematopoietic protein-tyrosine phosphatase | Protein-tyrosine phosphatase LC-PTP | Tyrosine-protein phosphatase non-receptor type 7 | Tyrosine-protein phosphatase non-receptor type 7 (HEPTP)
Type:Protein
Mol. Mass.:40530.79
Organism:Homo sapiens (Human)
Description:P35236
Residue:360
Sequence:
MVQAHGGRSRAQPLTLSLGAAMTQPPPEKTPAKKHVRLQERRGSNVALMLDVRSLGAVEP
ICSVNTPREVTLHFLRTAGHPLTRWALQRQPPSPKQLEEEFLKIPSNFVSPEDLDIPGHA
SKDRYKTILPNPQSRVCLGRAQSQEDGDYINANYIRGYDGKEKVYIATQGPMPNTVSDFW
EMVWQEEVSLIVMLTQLREGKEKCVHYWPTEEETYGPFQIRIQDMKECPEYTVRQLTIQY
QEERRSVKHILFSAWPDHQTPESAGPLLRLVAEVEESPETAAHPGPIVVHCSAGIGRTGC
FIATRIGCQQLKARGEVDILGIVCQLRLDRGGMIQTAEQYQFLHHTLALYAGQLPEEPSP
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  Blast E-value cutoff:
BDBM46207
n/a
NameBDBM46207
Synonyms:4-[[5-(4-bromophenyl)-2-furoyl]thiocarbamoylamino]benzoic acid | 4-[[5-(4-bromophenyl)furan-2-carbonyl]carbamothioylamino]benzoic acid | 4-[[5-(4-bromophenyl)furan-2-yl]carbonylcarbamothioylamino]benzoic acid | 4-[[[[[5-(4-bromophenyl)-2-furanyl]-oxomethyl]amino]-sulfanylidenemethyl]amino]benzoic acid | MLS-0383777.0001 | cid_1328767
TypeSmall organic molecule
Emp. Form.C19H13BrN2O4S
Mol. Mass.445.287
SMILESOC(=O)c1ccc(NC(=S)NC(=O)c2ccc(o2)-c2ccc(Br)cc2)cc1
Structure
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