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TargetGlutathione S-transferase Mu 1
LigandBDBM33107
Substrate/Competitorn/a
Meas. Tech.Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer)
EC50 3040±n/a nM
Citation PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Glutathione S-transferase Mu 1
Name:Glutathione S-transferase Mu 1
Synonyms:GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase
Type:PROTEIN
Mol. Mass.:25712.03
Organism:Homo sapiens (Human)
Description:ChEMBL_799596
Residue:218
Sequence:
MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNL
PYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEF
EKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPN
LKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
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  Blast E-value cutoff:
BDBM33107
n/a
NameBDBM33107
Synonyms:2-chloranyl-3-[[4-(diethylamino)phenyl]amino]naphthalene-1,4-dione | 2-chloro-3-[4-(diethylamino)anilino]-1,4-naphthoquinone | 2-chloro-3-[4-(diethylamino)anilino]naphthalene-1,4-dione | 2-chloro-3-{[4-(diethylamino)phenyl]amino}naphthoquinone | MLS000595078 | SMR000184814 | cid_1380424
TypeSmall organic molecule
Emp. Form.C20H19ClN2O2
Mol. Mass.354.83
SMILESCCN(CC)c1ccc(NC2=C(Cl)C(=O)c3ccccc3C2=O)cc1 |c:10|
Structure
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