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TargetMucolipin-3
LigandBDBM46826
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3)
EC50>29900±n/a nM
Citation PubChem, PC Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3) PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Mucolipin-3
Name:Mucolipin-3
Synonyms:MCLN3_HUMAN | MCOLN3 | MCOLN3 protein
Type:Enzyme Catalytic Domain
Mol. Mass.:64244.09
Organism:Homo sapiens (Human)
Description:Q8TDD5
Residue:553
Sequence:
MADPEVVVSSCSSHEEENRCNFNQQTSPSEELLLEDQMRRKLKFFFMNPCEKFWARGRKP
WKLAIQILKIAMVTIQLVLFGLSNQMVVAFKEENTIAFKHLFLKGYMDRMDDTYAVYTQS
DVYDQLIFAVNQYLQLYNVSVGNHAYENKGTKQSAMAICQHFYKRGNIYPGNDTFDIDPE
IETECFFVEPDEPFHIGTPAENKLNLTLDFHRLLTVELQFKLKAINLQTVRHQELPDCYD
FTLTITFDNKAHSGRIKISLDNDISIRECKDWHVSGSIQKNTHYMMIFDAFVILTCLVSL
ILCIRSVIRGLQLQQEFVNFFLLHYKKEVSVSDQMEFVNGWYIMIIISDILTIIGSILKM
EIQAKSLTSYDVCSILLGTSTMLVWLGVIRYLGFFAKYNLLILTLQAALPNVIRFCCCAA
MIYLGYCFCGWIVLGPYHDKFRSLNMVSECLFSLINGDDMFATFAKMQQKSYLVWLFSRI
YLYSFISLFIYMILSLFIALITDTYETIKQYQQDGFPETELRTFISECKDLPNSGKYRLE
DDPPVSLFCCCKK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM46826
n/a
NameBDBM46826
Synonyms:3-(3,5-dimethylphenyl)-2-(2-thienyl)thiazolidin-4-one | 3-(3,5-dimethylphenyl)-2-thiophen-2-yl-1,3-thiazolidin-4-one | 3-(3,5-dimethylphenyl)-2-thiophen-2-yl-4-thiazolidinone | MLS000078705 | SMR000034727 | cid_660804
TypeSmall organic molecule
Emp. Form.C15H15NOS2
Mol. Mass.289.416
SMILESCc1cc(C)cc(c1)N1C(SCC1=O)c1cccs1
Structure
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