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TargetMucolipin-3
LigandBDBM44578
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3)
EC50>29900±n/a nM
Citation PubChem, PC Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3) PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Mucolipin-3
Name:Mucolipin-3
Synonyms:MCLN3_HUMAN | MCOLN3 | MCOLN3 protein
Type:Enzyme Catalytic Domain
Mol. Mass.:64244.09
Organism:Homo sapiens (Human)
Description:Q8TDD5
Residue:553
Sequence:
MADPEVVVSSCSSHEEENRCNFNQQTSPSEELLLEDQMRRKLKFFFMNPCEKFWARGRKP
WKLAIQILKIAMVTIQLVLFGLSNQMVVAFKEENTIAFKHLFLKGYMDRMDDTYAVYTQS
DVYDQLIFAVNQYLQLYNVSVGNHAYENKGTKQSAMAICQHFYKRGNIYPGNDTFDIDPE
IETECFFVEPDEPFHIGTPAENKLNLTLDFHRLLTVELQFKLKAINLQTVRHQELPDCYD
FTLTITFDNKAHSGRIKISLDNDISIRECKDWHVSGSIQKNTHYMMIFDAFVILTCLVSL
ILCIRSVIRGLQLQQEFVNFFLLHYKKEVSVSDQMEFVNGWYIMIIISDILTIIGSILKM
EIQAKSLTSYDVCSILLGTSTMLVWLGVIRYLGFFAKYNLLILTLQAALPNVIRFCCCAA
MIYLGYCFCGWIVLGPYHDKFRSLNMVSECLFSLINGDDMFATFAKMQQKSYLVWLFSRI
YLYSFISLFIYMILSLFIALITDTYETIKQYQQDGFPETELRTFISECKDLPNSGKYRLE
DDPPVSLFCCCKK
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  Blast E-value cutoff:
BDBM44578
n/a
NameBDBM44578
Synonyms:1-(5-bromanylthiophen-2-yl)sulfonyl-4-methyl-piperidine | 1-(5-bromothiophen-2-yl)sulfonyl-4-methylpiperidine | 1-[(5-bromo-2-thienyl)sulfonyl]-4-methyl-piperidine | 1-[(5-bromo-2-thienyl)sulfonyl]-4-methylpiperidine | 1-[(5-bromo-2-thiophenyl)sulfonyl]-4-methylpiperidine | FLURANDRENOLIDE | MLS000069556 | MLS000099277 | SMR000058825 | SMR000073540 | cid_15209 | cid_893468
TypeSmall organic molecule
Emp. Form.C10H14BrNO2S2
Mol. Mass.324.258
SMILESCC1CCN(CC1)S(=O)(=O)c1ccc(Br)s1
Structure
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