| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Regulator of G-protein signaling 19 |
|---|
| Ligand | BDBM47698 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. |
|---|
| EC50 | >30000±n/a nM |
|---|
| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Regulator of G-protein signaling 19 |
|---|
| Name: | Regulator of G-protein signaling 19 |
|---|
| Synonyms: | G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19) |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 24631.38 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_86990435 |
|---|
| Residue: | 217 |
|---|
| Sequence: | MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
|
|
|
|---|
| BDBM47698 |
|---|
| n/a |
|---|
| Name | BDBM47698 |
|---|
| Synonyms: | 5-tert-butyl-3-[(2-chlorophenyl)methyl]-N-(2-morpholin-4-ylethyl)-[1,2,3]triazolo[4,5-d]pyrimidin-7-amine | 5-tert-butyl-3-[(2-chlorophenyl)methyl]-N-(2-morpholin-4-ylethyl)triazolo[4,5-d]pyrimidin-7-amine | 5-tert-butyl-3-[(2-chlorophenyl)methyl]-N-[2-(4-morpholinyl)ethyl]-7-triazolo[4,5-d]pyrimidinamine | MLS000034072 | SMR000007885 | [5-tert-Butyl-3-(2-chloro-benzyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-(2-morpholin-4-yl-ethyl)-amine | [5-tert-butyl-3-(2-chlorobenzyl)triazolo[4,5-d]pyrimidin-7-yl]-(2-morpholinoethyl)amine | cid_654918 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H28ClN7O |
|---|
| Mol. Mass. | 429.946 |
|---|
| SMILES | CC(C)(C)c1nc(NCCN2CCOCC2)c2nnn(Cc3ccccc3Cl)c2n1 |
|---|
| Structure | 
|
|---|
Search and Browse
