Ki Summary

Reaction Details

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Target

Regulator of G-protein signaling 19

Ligand

BDBM47701

Substrate/Competitor

n/a

Meas. Tech.

Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.

EC50

>30000±n/a nM

Citation

PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Regulator of G-protein signaling 19

Name:

Regulator of G-protein signaling 19

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

24631.38

Organism:

Homo sapiens (Human)

Description:

gi_86990435

Residue:

217

Sequence:

MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA

BDBM47701

n/a

Name

BDBM47701

Synonyms:

3-(2-hydroxy-3-phenoxypropyl)-5-[oxo-[(phenylmethyl)amino]methyl]-4-imidazolecarboxylic acid methyl ester | 5-(benzylcarbamoyl)-3-(2-hydroxy-3-phenoxy-propyl)imidazole-4-carboxylic acid methyl ester | MLS000082701 | SMR000046071 | cid_665038 | methyl 3-(2-oxidanyl-3-phenoxy-propyl)-5-[(phenylmethyl)carbamoyl]imidazole-4-carboxylate | methyl 5-(benzylcarbamoyl)-3-(2-hydroxy-3-phenoxypropyl)imidazole-4-carboxylate

Type

Small organic molecule

Emp. Form.

C22H23N3O5

Mol. Mass.

409.4351

SMILES

COC(=O)c1c(ncn1CC(O)COc1ccccc1)C(=O)NCc1ccccc1

Structure