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TargetRegulator of G-protein signaling 16
LigandBDBM47765
Substrate/Competitorn/a
Meas. Tech.Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50>30000±n/a nM
Citation PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 16
Name:Regulator of G-protein signaling 16
Synonyms:RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:Enzyme Catalytic Domain
Mol. Mass.:22748.87
Organism:Homo sapiens (Human)
Description:gi_156416009
Residue:202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
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BDBM47765
n/a
NameBDBM47765
Synonyms:MLS000677175 | N-(dibenzylcarbamothioyl)-2-methylpropanamide | N-(dibenzylthiocarbamoyl)-2-methyl-propionamide | N-[(dibenzylamino)carbonothioyl]-2-methylpropanamide | N-[[bis(phenylmethyl)amino]-sulfanylidenemethyl]-2-methylpropanamide | N-[bis(phenylmethyl)carbamothioyl]-2-methyl-propanamide | SMR000270987 | cid_801325
TypeSmall organic molecule
Emp. Form.C19H22N2OS
Mol. Mass.326.456
SMILESCC(C)C(=O)NC(=S)N(Cc1ccccc1)Cc1ccccc1
Structure
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