Reaction Details |
| Report a problem with these data |
Target | Regulator of G-protein signaling 16 |
---|
Ligand | BDBM34849 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. |
---|
EC50 | 16000±n/a nM |
---|
Citation | PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID] |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
Regulator of G-protein signaling 16 |
---|
Name: | Regulator of G-protein signaling 16 |
Synonyms: | RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 22748.87 |
Organism: | Homo sapiens (Human) |
Description: | gi_156416009 |
Residue: | 202 |
Sequence: | MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
|
|
|
BDBM34849 |
---|
n/a |
---|
Name | BDBM34849 |
Synonyms: | 6-fluoranyl-2-(2-methylphenyl)-1,2-benzothiazol-3-one | 6-fluoro-2-(2-methylphenyl)-1,2-benzisothiazol-3(2H)-one | 6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-one | 6-fluoro-2-(o-tolyl)-1,2-benzothiazol-3-one | MLS000729299 | SMR000307577 | cid_1510379 |
Type | Small organic molecule |
Emp. Form. | C14H10FNOS |
Mol. Mass. | 259.299 |
SMILES | Cc1ccccc1-n1sc2cc(F)ccc2c1=O |
Structure |
|