| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 16 |
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| Ligand | BDBM47798 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. |
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| EC50 | 1630±n/a nM |
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| Citation |  PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Regulator of G-protein signaling 16 |
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| Name: | Regulator of G-protein signaling 16 |
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| Synonyms: | RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 22748.87 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_156416009 |
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| Residue: | 202 |
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| Sequence: | MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
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| BDBM47798 |
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| n/a |
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| Name | BDBM47798 |
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| Synonyms: | 4-chloranyl-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N-methyl-1,3,5-triazin-2-amine | 4-chloro-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N-methyl-1,3,5-triazin-2-amine | 4-chloro-6-[(4,6-dimethyl-2-pyrimidinyl)thio]-N-methyl-1,3,5-triazin-2-amine | MLS000707335 | SMR000288800 | [4-chloro-6-[(4,6-dimethylpyrimidin-2-yl)thio]-s-triazin-2-yl]-methyl-amine | cid_1087037 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H11ClN6S |
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| Mol. Mass. | 282.753 |
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| SMILES | CNc1nc(Cl)nc(Sc2nc(C)cc(C)n2)n1 |
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| Structure | 
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