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TargetDual specificity protein phosphatase (VHR)
LigandBDBM46224
Substrate/Competitorn/a
Meas. Tech.SAR VHR1 absorbance Assay for In Vitro dose response studies.
IC50 3620±n/a nM
Citation PubChem PC SAR VHR1 absorbance Assay for In Vitro dose response studies. PubChem Bioassay (2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase (VHR)
Name:Dual specificity protein phosphatase 3
Synonyms:Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR
Type:Hydrolase
Mol. Mass.:20480.58
Organism:Homo sapiens (Human)
Description:n/a
Residue:185
Sequence:
MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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BDBM46224
n/a
NameBDBM46224
Synonyms:2-[2-bromanyl-4-[(Z)-[2-[(4-ethylphenyl)amino]-4-oxidanylidene-1,3-thiazol-5-ylidene]methyl]-6-methoxy-phenoxy]ethanoic acid | 2-[2-bromo-4-[(Z)-[2-(4-ethylanilino)-4-keto-2-thiazolin-5-ylidene]methyl]-6-methoxy-phenoxy]acetic acid | 2-[2-bromo-4-[(Z)-[2-(4-ethylanilino)-4-oxo-1,3-thiazol-5-ylidene]methyl]-6-methoxyphenoxy]acetic acid | 2-[2-bromo-4-[(Z)-[2-(4-ethylanilino)-4-oxo-5-thiazolylidene]methyl]-6-methoxyphenoxy]acetic acid | MLS-0343544.0001 | cid_5765581
TypeSmall organic molecule
Emp. Form.C21H19BrN2O5S
Mol. Mass.491.355
SMILESCCc1ccc(NC2=NC(=O)C(S2)=Cc2cc(Br)c(OCC(O)=O)c(OC)c2)cc1 |w:13.14,t:7|
Structure
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