Reaction Details |
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Target | Regulator of G-protein signaling 4 |
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Ligand | BDBM47695 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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EC50 | 30000±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 4 |
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Name: | Regulator of G-protein signaling 4 |
Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
Type: | Enzyme |
Mol. Mass.: | 23263.51 |
Organism: | Homo sapiens (Human) |
Description: | P49798 |
Residue: | 205 |
Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47695 |
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n/a |
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Name | BDBM47695 |
Synonyms: | 2-(N-[2-(1-benzotriazolyl)-1-oxoethyl]-2-methoxyanilino)-N-(2-methylbutan-2-yl)-2-(1-methyl-2-pyrrolyl)acetamide | 2-(N-[2-(benzotriazol-1-yl)acetyl]-2-methoxyanilino)-N-(2-methylbutan-2-yl)-2-(1-methylpyrrol-2-yl)acetamide | 2-[(2-Benzotriazol-1-yl-acetyl)-(2-methoxy-phenyl)-amino]-N-(1,1-dimethyl-propyl)-2-(1-methyl-1H-pyrrol-2-yl)-acetamide | 2-[2-(benzotriazol-1-yl)ethanoyl-(2-methoxyphenyl)amino]-N-(2-methylbutan-2-yl)-2-(1-methylpyrrol-2-yl)ethanamide | MLS000074185 | N-tert-amyl-2-(N-[2-(benzotriazol-1-yl)acetyl]-2-methoxy-anilino)-2-(1-methylpyrrol-2-yl)acetamide | SMR000004342 | cid_646963 |
Type | Small organic molecule |
Emp. Form. | C27H32N6O3 |
Mol. Mass. | 488.5814 |
SMILES | CCC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccccc1OC)c1cccn1C |
Structure |
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