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Targetregulator of G-protein signaling 4
LigandBDBM47697
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao.
EC50 30000±n/a nM
Citation PubChem PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay (2009)[AID]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4 (RGS4)
Synonyms:RGP4 | RGS4
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47697
n/a
NameBDBM47697
Synonyms:MLS000071118 | SMR000003789 | [2-(2,3-dihydro-1H-inden-5-ylamino)-3-pyridinyl]-(4-morpholinyl)methanone | [2-(2,3-dihydro-1H-inden-5-ylamino)pyridin-3-yl]-morpholin-4-yl-methanone | [2-(2,3-dihydro-1H-inden-5-ylamino)pyridin-3-yl]-morpholin-4-ylmethanone | [2-(Indan-5-ylamino)-pyridin-3-yl]-morpholin-4-yl-methanone | [2-(indan-5-ylamino)-3-pyridyl]-morpholino-methanone | cid_651142
TypeSmall organic molecule
Emp. Form.C19H21N3O2
Mol. Mass.323.3889
SMILESO=C(N1CCOCC1)c1cccnc1Nc1ccc2CCCc2c1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: