Reaction Details |
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Target | Regulator of G-protein signaling 4 |
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Ligand | BDBM47703 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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EC50 | 30000±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 4 |
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Name: | Regulator of G-protein signaling 4 |
Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
Type: | Enzyme |
Mol. Mass.: | 23263.51 |
Organism: | Homo sapiens (Human) |
Description: | P49798 |
Residue: | 205 |
Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47703 |
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n/a |
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Name | BDBM47703 |
Synonyms: | 2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-(4-tert-butylanilino)-2-oxoethyl] ester | 2,3-dihydro-p-dioxin-5-carboxylic acid [2-(4-tert-butylanilino)-2-keto-ethyl] ester | MLS000082235 | SMR000061029 | [2-(4-tert-butylanilino)-2-oxoethyl] 2,3-dihydro-1,4-dioxine-5-carboxylate | [2-[(4-tert-butylphenyl)amino]-2-oxidanylidene-ethyl] 2,3-dihydro-1,4-dioxine-5-carboxylate | cid_2337962 |
Type | Small organic molecule |
Emp. Form. | C17H21NO5 |
Mol. Mass. | 319.3523 |
SMILES | CC(C)(C)c1ccc(NC(=O)COC(=O)C2=COCCO2)cc1 |t:15| |
Structure |
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