| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 4 |
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| Ligand | BDBM40034 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 4 |
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| Name: | Regulator of G-protein signaling 4 |
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| Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23263.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49798 |
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| Residue: | 205 |
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| Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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| BDBM40034 |
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| n/a |
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| Name | BDBM40034 |
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| Synonyms: | MLS000093573 | N-(3-keto-4-methyl-1,4-benzothiazin-6-yl)-4-piperidino-piperidine-1-carboxamide | N-(4-methyl-3-oxidanylidene-1,4-benzothiazin-6-yl)-4-piperidin-1-yl-piperidine-1-carboxamide | N-(4-methyl-3-oxo-1,4-benzothiazin-6-yl)-4-(1-piperidinyl)-1-piperidinecarboxamide | N-(4-methyl-3-oxo-1,4-benzothiazin-6-yl)-4-piperidin-1-ylpiperidine-1-carboxamide | N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-6-yl)-1,4'-bipiperidine-1'-carboxamide | SMR000029191 | cid_3241667 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H28N4O2S |
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| Mol. Mass. | 388.527 |
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| SMILES | CN1C(=O)CSc2ccc(NC(=O)N3CCC(CC3)N3CCCCC3)cc12 |
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| Structure | 
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