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TargetRegulator of G-protein signaling 4
LigandBDBM47705
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao.
EC50 30000±n/a nM
Citation PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4
Synonyms:RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47705
n/a
NameBDBM47705
Synonyms:1-[2-(difluoromethoxy)-5-methyl-phenyl]-3-(2,4-dimethoxyphenyl)urea | 1-[2-(difluoromethoxy)-5-methylphenyl]-3-(2,4-dimethoxyphenyl)urea | 1-[2-[bis(fluoranyl)methoxy]-5-methyl-phenyl]-3-(2,4-dimethoxyphenyl)urea | MLS000097201 | N-[2-(difluoromethoxy)-5-methylphenyl]-N'-(2,4-dimethoxyphenyl)urea | SMR000076793 | cid_2208379
TypeSmall organic molecule
Emp. Form.C17H18F2N2O4
Mol. Mass.352.3326
SMILESCOc1ccc(NC(=O)Nc2cc(C)ccc2OC(F)F)c(OC)c1
Structure
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