| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 4 |
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| Ligand | BDBM47709 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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| EC50 | 60±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 4 |
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| Name: | Regulator of G-protein signaling 4 |
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| Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23263.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49798 |
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| Residue: | 205 |
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| Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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| BDBM47709 |
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| n/a |
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| Name | BDBM47709 |
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| Synonyms: | 9-(2-thienyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one | 9-(2-thienyl)-5,6,7,9-tetrahydro[1,2,4]triazolo[5,1-b]quinazolin-8(4H)-one | 9-thiophen-2-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one | MLS000088907 | SMR000073127 | cid_5711559 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H12N4OS |
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| Mol. Mass. | 272.326 |
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| SMILES | O=C1CCCC2=Nc3ncnn3C(C12)c1cccs1 |t:5| |
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| Structure | 
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