| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 4 |
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| Ligand | BDBM47722 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 4 |
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| Name: | Regulator of G-protein signaling 4 |
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| Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23263.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49798 |
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| Residue: | 205 |
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| Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
|
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|
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| BDBM47722 |
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| n/a |
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| Name | BDBM47722 |
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| Synonyms: | 5-cyano-4-ethyl-2-methyl-N-phenyl-6-sulfanylidene-1H-pyridine-3-carboxamide | 5-cyano-4-ethyl-2-methyl-N-phenyl-6-thioxo-1,6-dihydro-3-pyridinecarboxamide | 5-cyano-4-ethyl-2-methyl-N-phenyl-6-thioxo-1H-pyridine-3-carboxamide | MLS000532290 | SMR000137229 | cid_789551 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H15N3OS |
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| Mol. Mass. | 297.375 |
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| SMILES | CCc1c(C#N)c(=S)[nH]c(C)c1C(=O)Nc1ccccc1 |
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| Structure | 
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