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TargetZinc finger protein mex-5
LigandBDBM52079
Substrate/Competitorn/a
Meas. Tech.Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50 12226±n/a nM
Citation PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Zinc finger protein mex-5
Name:Zinc finger protein mex-5
Synonyms:MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:Enzyme Catalytic Domain
Mol. Mass.:52832.78
Organism:Caenorhabditis elegans
Description:gi_55976631
Residue:468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
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  Blast E-value cutoff:
BDBM52079
n/a
NameBDBM52079
Synonyms:(5,5-diketo-6H-benzo[c][1,2]benzothiazin-9-yl)amine | 5,5-bis(oxidanylidene)-6H-benzo[c][1,2]benzothiazin-9-amine | 5,5-dioxo-6H-benzo[c][1,2]benzothiazin-9-amine | 9,9-Dioxo-9,10-dihydro-9lambda*6*-thia-10-aza-phenanthren-3-ylamine | MLS000073006 | SMR000010061 | cid_653405
TypeSmall organic molecule
Emp. Form.C12H10N2O2S
Mol. Mass.246.285
SMILESNc1ccc2NS(=O)(=O)c3ccccc3-c2c1
Structure
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