Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM52472

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

300000±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52472

n/a

Name

BDBM52472

Synonyms:

MLS000402404 | N-[(3-methyl-1-phenyl-5-pyrrolidin-1-yl-pyrazol-4-yl)methylideneamino]-2-pyridin-3-yl-quinoline-4-carboxamide | N-[(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]-2-pyridin-3-ylquinoline-4-carboxamide | N-[(3-methyl-1-phenyl-5-pyrrolidino-pyrazol-4-yl)methyleneamino]-2-(3-pyridyl)cinchoninamide | N-[[3-methyl-1-phenyl-5-(1-pyrrolidinyl)-4-pyrazolyl]methylideneamino]-2-(3-pyridinyl)-4-quinolinecarboxamide | SMR000262226 | cid_2328705

Type

Small organic molecule

Emp. Form.

C30H27N7O

Mol. Mass.

501.5817

SMILES

Cc1nn(c(N2CCCC2)c1C=NNC(=O)c1cc(nc2ccccc12)-c1cccnc1)-c1ccccc1 |w:12.14|

Structure