Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM52477

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

300000±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52477

n/a

Name

BDBM52477

Synonyms:

5-[2,5-dimethyl-3-[2-[2-(tosylamino)acetyl]oxyacetyl]pyrrol-1-yl]benzene-1,3-dicarboxylic acid dimethyl ester | 5-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]-1-oxoethoxy]-1-oxoethyl]-1-pyrrolyl]benzene-1,3-dicarboxylic acid dimethyl ester | MLS000393629 | SMR000247859 | cid_3494085 | dimethyl 5-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]acetyl]oxyacetyl]pyrrol-1-yl]benzene-1,3-dicarboxylate | dimethyl 5-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]ethanoyloxy]ethanoyl]pyrrol-1-yl]benzene-1,3-dicarboxylate

Type

Small organic molecule

Emp. Form.

C27H28N2O9S

Mol. Mass.

556.584

SMILES

COC(=O)c1cc(cc(c1)-n1c(C)cc(C(=O)COC(=O)CNS(=O)(=O)c2ccc(C)cc2)c1C)C(=O)OC

Structure