Ki Summary

Reaction Details

Report a problem with these data

Target

Zinc finger protein mex-5

Ligand

BDBM52478

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

14647±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52478

n/a

Name

BDBM52478

Synonyms:

3-(1,3-benzothiazol-2-ylsulfanyl)-N'-[(Z)-(2-oxidanylidenenaphthalen-1-ylidene)methyl]propanehydrazide | 3-(1,3-benzothiazol-2-ylsulfanyl)-N'-[(Z)-(2-oxonaphthalen-1-ylidene)methyl]propanehydrazide | 3-(1,3-benzothiazol-2-ylthio)-N'-[(Z)-(2-keto-1-naphthylidene)methyl]propionohydrazide | 3-(1,3-benzothiazol-2-ylthio)-N'-[(Z)-(2-oxo-1-naphthalenylidene)methyl]propanehydrazide | 3-(Benzothiazol-2-ylsulfanyl)-propionic acid [1-(2-hydroxy-naphthalen-1-yl)-meth-(E)-ylidene]-hydrazide | MLS000591355 | SMR000218975 | cid_6504438

Type

Small organic molecule

Emp. Form.

C21H17N3O2S2

Mol. Mass.

407.509

SMILES

Oc1ccc2ccccc2c1C=NNC(=O)CCSc1nc2ccccc2s1 |w:12.14|

Structure