Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM52480

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

300000±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52480

n/a

Name

BDBM52480

Synonyms:

2-[2-azanylidene-3-[(4-chlorophenyl)methyl]benzimidazol-1-yl]-1-(4-nitrophenyl)ethanone;hydrobromide | 2-[3-(4-Chloro-benzyl)-2-imino-2,3-dihydro-benzoimidazol-1-yl]-1-(4-nitro-phenyl)-ethanone | 2-[3-(4-chlorobenzyl)-2-imino-benzimidazol-1-yl]-1-(4-nitrophenyl)ethanone;hydrobromide | 2-[3-[(4-chlorophenyl)methyl]-2-imino-1-benzimidazolyl]-1-(4-nitrophenyl)ethanone;hydrobromide | 2-[3-[(4-chlorophenyl)methyl]-2-iminobenzimidazol-1-yl]-1-(4-nitrophenyl)ethanone;hydrobromide | MLS000588756 | SMR000212362 | cid_15944760

Type

Small organic molecule

Emp. Form.

C22H17ClN4O3

Mol. Mass.

420.848

SMILES

[O-][N+](=O)c1ccc(cc1)C(=O)Cn1c2ccccc2n(Cc2ccc(Cl)cc2)c1=N

Structure