Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM51083

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

56744±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM51083

n/a

Name

BDBM51083

Synonyms:

(4Z)-2-(4-fluorophenyl)-4-[(3-methyl-1-phenyl-5-pyrrolidin-1-yl-pyrazol-4-yl)methylidene]-1,3-oxazol-5-one | (4Z)-2-(4-fluorophenyl)-4-[(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylidene]-1,3-oxazol-5-one | (4Z)-2-(4-fluorophenyl)-4-[(3-methyl-1-phenyl-5-pyrrolidino-pyrazol-4-yl)methylene]-2-oxazolin-5-one | (4Z)-2-(4-fluorophenyl)-4-[[3-methyl-1-phenyl-5-(1-pyrrolidinyl)-4-pyrazolyl]methylidene]-5-oxazolone | MLS000391676 | SMR000260711 | cid_2327951

Type

Small organic molecule

Emp. Form.

C24H21FN4O2

Mol. Mass.

416.4475

SMILES

Cc1nn(c(N2CCCC2)c1\C=C1/N=C(OC1=O)c1ccc(F)cc1)-c1ccccc1 |c:15|

Structure