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TargetZinc finger protein mex-5
LigandBDBM52485
Substrate/Competitorn/a
Meas. Tech.Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50 12820±n/a nM
Citation PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Zinc finger protein mex-5
Name:Zinc finger protein mex-5
Synonyms:MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:Enzyme Catalytic Domain
Mol. Mass.:52832.78
Organism:Caenorhabditis elegans
Description:gi_55976631
Residue:468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
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  Blast E-value cutoff:
BDBM52485
n/a
NameBDBM52485
Synonyms:5-(4-fluorophenyl)-7-(2-furanyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine | 5-(4-fluorophenyl)-7-(2-furyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine | 5-(4-fluorophenyl)-7-(2-furyl)-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidine | 5-(4-fluorophenyl)-7-(furan-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine | MLS000626960 | SMR000272093 | cid_5736758
TypeSmall organic molecule
Emp. Form.C15H11FN4O
Mol. Mass.282.2724
SMILESFc1ccc(cc1)C1=Nc2ncnn2C(C1)c1ccco1 |t:8|
Structure
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