Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM52492

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

300000±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52492

n/a

Name

BDBM52492

Synonyms:

(E)-1-(2,4-dimethoxyphenyl)-3-(3-nitro-4-piperidin-1-yl-phenyl)prop-2-en-1-one | (E)-1-(2,4-dimethoxyphenyl)-3-(3-nitro-4-piperidin-1-ylphenyl)prop-2-en-1-one | (E)-1-(2,4-dimethoxyphenyl)-3-(3-nitro-4-piperidino-phenyl)prop-2-en-1-one | (E)-1-(2,4-dimethoxyphenyl)-3-[3-nitro-4-(1-piperidinyl)phenyl]-2-propen-1-one | MLS000390406 | SMR000255373 | cid_15945163

Type

Small organic molecule

Emp. Form.

C22H24N2O5

Mol. Mass.

396.4364

SMILES

COc1ccc(C(=O)\C=C\c2ccc(N3CCCCC3)c(c2)[N+]([O-])=O)c(OC)c1

Structure