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TargetZinc finger protein mex-5
LigandBDBM52501
Substrate/Competitorn/a
Meas. Tech.Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50 300000±n/a nM
Citation PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Zinc finger protein mex-5
Name:Zinc finger protein mex-5
Synonyms:MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:Enzyme Catalytic Domain
Mol. Mass.:52832.78
Organism:Caenorhabditis elegans
Description:gi_55976631
Residue:468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
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  Blast E-value cutoff:
BDBM52501
n/a
NameBDBM52501
Synonyms:1-phenyl-6-(pyrimidin-2-ylsulfanylmethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one | 1-phenyl-6-[(2-pyrimidinylthio)methyl]-2H-pyrazolo[3,4-d]pyrimidin-4-one | 1-phenyl-6-[(2-pyrimidylthio)methyl]-2H-pyrazolo[3,4-d]pyrimidin-4-one | MLS000417818 | SMR000243299 | cid_701317
TypeSmall organic molecule
Emp. Form.C16H12N6OS
Mol. Mass.336.371
SMILESO=c1[nH]c(CSc2ncccn2)nc2n(ncc12)-c1ccccc1
Structure
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