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TargetDual specificity protein phosphatase 6
LigandBDBM32047
Substrate/Competitorn/a
Meas. Tech.MKP-3 in vitro HTS assay
IC50 10000±n/a nM
Citation PubChem, PC MKP-3 in vitro HTS assay PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase 6
Name:Dual specificity protein phosphatase 6
Synonyms:DUS6_RAT | Dusp6 | MAP kinase phosphatase 3 | MKP-3 | Mitogen-activated protein kinase phosphatase 3 | Mkp3
Type:Enzyme
Mol. Mass.:42303.19
Organism:Rattus norvegicus
Description:gi_16758752
Residue:381
Sequence:
MIDTLRPVPFASEMAISKTVAWLNEQLELGNEQLLLMDCRPQELYESSHIESAINVAIPG
IMLRRLQKGNLPVRALFTRCEDRDRFTRRCGTDTVVLYDENSSDWNENTGGESVLGLLLK
KLKDEGCRAFYLEGGFSKFQAEFALHCETNLDGSCSSSSPPLPVLGLGGLRISSDSSSDI
ESDLDRDPNSATDSDGSPLSNSQPSFPVEILPFLYLGCAKDSTNLDVLEEFGIKYILNVT
PNLPNLFENAGEFKYKQIPISDHWSQNLSQFFPEAISFIDEARGKNCGVLVHCLAGISRS
VTVTVAYLMQKLNLSMNDAYDIVKMKKSNISPNFNFMGQLLDFERTLGLSSPCDNRVPAQ
QLYFTAPSNQNVYQVDSLQST
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  Blast E-value cutoff:
BDBM32047
n/a
NameBDBM32047
Synonyms:(5-amino-6-quinolyl)amine | MLS000036429 | SMR000015817 | cid_426874 | quinoline-5,6-diamine
TypeSmall organic molecule
Emp. Form.C9H9N3
Mol. Mass.159.1879
SMILESNc1ccc2ncccc2c1N
Structure
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