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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Dual specificity protein phosphatase 6 | ||
| Ligand | BDBM31754 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | MKP-3 in vitro HTS assay | ||
| IC50 | 11000±n/a nM | ||
| Citation |  PubChem, PC MKP-3 in vitro HTS assay PubChem Bioassay(2009)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Dual specificity protein phosphatase 6 | |||
| Name: | Dual specificity protein phosphatase 6 | ||
| Synonyms: | DUS6_RAT | Dusp6 | MAP kinase phosphatase 3 | MKP-3 | Mitogen-activated protein kinase phosphatase 3 | Mkp3 | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 42303.19 | ||
| Organism: | Rattus norvegicus | ||
| Description: | gi_16758752 | ||
| Residue: | 381 | ||
| Sequence: |
| ||
| BDBM31754 | |||
| n/a | |||
| Name | BDBM31754 | ||
| Synonyms: | MLS-0010366.0001 | N-(5-phenyl-1,2,4-thiadiazol-3-yl)-2-[(5-phenyl-3-thiazolo[2,3-c][1,2,4]triazolyl)thio]acetamide | N-(5-phenyl-1,2,4-thiadiazol-3-yl)-2-[(5-phenyl-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl)sulfanyl]acetamide | N-(5-phenyl-1,2,4-thiadiazol-3-yl)-2-[(5-phenyl-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl)sulfanyl]ethanamide | N-(5-phenyl-1,2,4-thiadiazol-3-yl)-2-[(5-phenylthiazolo[2,3-c][1,2,4]triazol-3-yl)thio]acetamide | cid_1589738 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C20H14N6OS3 | ||
| Mol. Mass. | 450.56 | ||
| SMILES | O=C(CSc1nnc2scc(-c3ccccc3)n12)Nc1nsc(n1)-c1ccccc1 | ||
| Structure | 
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