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TargetCell division control protein 42 homolog
LigandBDBM54555
Substrate/Competitorn/a
Meas. Tech.Oxadiazole SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
Ki 280±n/a nM
Citation PubChem, PC Oxadiazole SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM54555
n/a
NameBDBM54555
Synonyms:1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-propanone | 1-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one | 1-[4-(2,5-dimethylphenyl)piperazino]-3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one | KUC103366N | UNM-0000306076 | cid_42596904
TypeSmall organic molecule
Emp. Form.C23H25FN4O2
Mol. Mass.408.4686
SMILESCc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCc1nc(no1)-c1cccc(F)c1
Structure
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