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TargetCell division control protein 42 homolog
LigandBDBM54607
Substrate/Competitorn/a
Meas. Tech.Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
Ki 10±n/a nM
Citation PubChem, PC Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM54607
n/a
NameBDBM54607
Synonyms:4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimethyl-aniline | 4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimethylaniline | UNM-0000305845 | [4-(2,5-diphenyl-2-pyrazolin-3-yl)phenyl]-dimethyl-amine | cid_2729182
TypeSmall organic molecule
Emp. Form.C23H23N3
Mol. Mass.341.4488
SMILESCN(C)c1ccc(cc1)C1CC(=NN1c1ccccc1)c1ccccc1 |c:12|
Structure
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