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TargetRas-related C3 botulinum toxin substrate 1
LigandBDBM54562
Substrate/Competitorn/a
Meas. Tech.Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype
Ki 170±n/a nM
Citation PubChem, PC Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related C3 botulinum toxin substrate 1
Name:Ras-related C3 botulinum toxin substrate 1
Synonyms:RAC1_MOUSE | Rac1 | Rac1 protein
Type:PROTEIN
Mol. Mass.:21455.91
Organism:Mus musculus
Description:EBI_101485
Residue:192
Sequence:
MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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BDBM54562
n/a
NameBDBM54562
Synonyms:3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-1-propanone | 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-1-[4-(2,5-dimethylphenyl)piperazin-1-yl]propan-1-one | 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-1-[4-(2,5-dimethylphenyl)piperazino]propan-1-one | KUC103373N | UNM-0000306083 | cid_42596910
TypeSmall organic molecule
Emp. Form.C23H25ClN4O2
Mol. Mass.424.923
SMILESCc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCc1nc(no1)-c1ccc(Cl)cc1
Structure
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