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TargetGTPase KRas [1-37]
LigandBDBM54607
Substrate/Competitorn/a
Meas. Tech.Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Ras wildtype
Ki 10±n/a nM
Citation PubChem, PC Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Ras wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
GTPase KRas [1-37]
Name:GTPase KRas [1-37]
Synonyms:ras protein
Type:Enzyme Catalytic Domain
Mol. Mass.:4034.04
Organism:Homo sapiens (Human)
Description:gi_190938
Residue:37
Sequence:
MTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIE
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  Blast E-value cutoff:
BDBM54607
n/a
NameBDBM54607
Synonyms:4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimethyl-aniline | 4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimethylaniline | UNM-0000305845 | [4-(2,5-diphenyl-2-pyrazolin-3-yl)phenyl]-dimethyl-amine | cid_2729182
TypeSmall organic molecule
Emp. Form.C23H23N3
Mol. Mass.341.4488
SMILESCN(C)c1ccc(cc1)C1CC(=NN1c1ccccc1)c1ccccc1 |c:12|
Structure
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